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1

Discovery of a Potent and Selective Prostaglandin D 2 Receptor Antagonist, [(3 R )-4-(4-Chloro- benzyl)-7-fluoro-5-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[ b ]indol-3-yl]-acetic Acid (MK-0524) †

Sturino, Claudio F., O'Neill, Gary, Lachance, Nicolas, Boyd, Michael, Berthelette, Carl, Labelle, Marc, Li, Lianhai, Roy, Bruno, Scheigetz, John, Tsou, Nancy, Aubin, Yves, Bateman, Kevin P., Chauret,

Journal:

Journal of Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 165 KB

english, 2007

2

Development of 2,3-dihydro-6-(3-phenoxypropyl)-2-(2-phenylethyl)-5-benzofuranol (L-670,630) as a potent and orally active inhibitor of 5-lipoxygenase

Lau, Cheuk K., Belanger, Patrice C., Dufresne, Claude, Scheigetz, John, Therien, Michel, Fitzsimmons, Brian, Young, Robert N., Ford-Hutchinson, Anthony W., Riendeau, Denis

Journal:

Journal of Medicinal Chemistry

Year:

1992

Language:

english

File:

PDF, 2.66 MB

english, 1992

3

ChemInform Abstract: Synthesis of Fluorescein Phosphorotriesters Using Photolabile Protecting Groups.

John Scheigetz, Bruno Roy

Journal:

Year:

2000

File:

PDF, 27 KB

2000

4

ChemInform Abstract: Synthesis of N-Aminoindole Ureas from Ethyl 1-Amino-6-(trifluoromethyl)-1H-indole-3-carboxylate.

Michel Belley, John Scheigetz, Pascal Dube, Sarah Dolman

Journal:

Year:

2001

File:

PDF, 30 KB

2001

5

Synthesis and characterization of tritium labeled 2,3,4,9-tetrahydro-1H-carbazoles as potent DP receptor antagonists

Carl Berthelette, Michael J. Boyd, Nicolas Lachance, Bruno Roy, Claudio F. Sturino, John Scheigetz, Robert J. Zamboni

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

2004

Language:

english

File:

PDF, 109 KB

english, 2004

6

Base-catalyzed deuterium and tritium labelling of 1-biphenyl-4-ylpropane-1,2-dione and deuteration of aryl methyl ketones

Carl Berthelette, John Scheigetz

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

2004

Language:

english

File:

PDF, 78 KB

english, 2004

7

Base-catalyzed deuterium and tritium labeling of aryl methyl sulfones

John Scheigetz, Carl Berthelette, Chun Li, Robert J. Zamboni

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

2004

Language:

english

File:

PDF, 118 KB

english, 2004

8

Discovery of a substituted 8-arylquinoline series of PDE4 inhibitors: Structure–activity relationship, optimization, and identification of a highly potent, well tolerated, PDE4 inhibitor

Dwight Macdonald, Anthony Mastracchio, Hélène Perrier, Daniel Dubé, Michel Gallant, Patrick Lacombe, Denis Deschênes, Bruno Roy, John Scheigetz, Kevin Bateman, Chun Li, Laird A. Trimble, Stephen Day,

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 155 KB

english, 2005

9

Investigation of ketone warheads as alternatives to the nitrile for preparation of potent and selective cathepsin K inhibitors

Michael J. Boyd, Sheldon N. Crane, Joël Robichaud, John Scheigetz, W. Cameron Black, Nathalie Chauret, Qingping Wang, Frédéric Massé, Renata M. Oballa

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2009

Language:

english

File:

PDF, 163 KB

english, 2009

10

Formation of a novel thiopyranoindole ring system

John H. Hutchinson, Ernie J. McEachern, John Scheigetz, Dwight Macdonald, Michel Thérien

Journal:

Tetrahedron Letters

Year:

1992

Language:

english

File:

PDF, 254 KB

english, 1992

11

Identification of an indole series of prostaglandin D2 receptor antagonists

Claudio F. Sturino, Nicolas Lachance, Michael Boyd, Carl Berthelette, Marc Labelle, Lianhai Li, Bruno Roy, John Scheigetz, Nancy Tsou, Christine Brideau, Elizabeth Cauchon, Marie-Claude Carriere, Dani

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2006

Language:

english

File:

PDF, 163 KB

english, 2006

12

Novel caged fluorescein diphosphates as photoactivatable substrates for protein tyrosine phosphatases

Qingping Wang, John Scheigetz, Bruno Roy, Chidambaram Ramachandran, Michael J Gresser

Journal:

Biochimica et Biophysica Acta (BBA) - Proteins and Proteomics

Year:

2002

Language:

english

File:

PDF, 349 KB

english, 2002

13

Reductive deoxygenation of aryl aldehydes and ketones by tert-butylamine-borane and aluminum chloride

Lau, Cheuk K., Tardif, Sylvie, Dufresne, Claude, Scheigetz, John

Journal:

Journal of Organic Chemistry

Year:

1989

Language:

english

File:

PDF, 467 KB

english, 1989

14

Synthesis and stereochemistry of 11-substituted 5,6,7,8,9,10-hexahydro-6,9-methanobenzocyclooctenes

Belanger, Patrice C., Young, Robert N., Scheigetz, John S., Dufresne, Claude, Springer, James P.

Journal:

Journal of Organic Chemistry

Year:

1982

Language:

english

File:

PDF, 1.34 MB

english, 1982

15

Fluorescein monophosphates as fluorogenic substrates for protein tyrosine phosphatases

Qingping Wang, John Scheigetz, Michael Gilbert, Jamie Snider, Chidambaram Ramachandran

Journal:

Biochimica et Biophysica Acta (BBA) - Protein Structure and Molecular Enzymology

Year:

1999

Language:

english

File:

PDF, 374 KB

english, 1999

16

Reductive deoxygenation of aryl aldehydes and ketones and benzylic, allylic, and tertiary alcohols by zinc iodide-sodium cyanoborohydride

Lau, C. K., Dufresne, Claude, Belanger, Patrice C., Pietre, Sylvie, Scheigetz, John

Journal:

Journal of Organic Chemistry

Year:

1986

Language:

english

File:

PDF, 631 KB

english, 1986

17

ortho -Specific alkylation of phenols via 1,3,2-benzodioxaborins

Lau, Cheuk K., Williams, Haydn W.R., Tardiff, Sylvie, Dufresne, Claude, Scheigetz, John, Bélanger, Patrice C.

Journal:

Canadian Journal of Chemistry

Year:

1989

Language:

english

File:

PDF, 266 KB

english, 1989

18

A SYNTHESIS OF 4-α-GUANIDINO-2-DEOXY-2,3-DIDEHYDRO N-ACETYLNEURAMINIC ACID

Scheigetz, John, Zamboni, Robert, Bernstein, Michael A., Roy, Bruno

Journal:

Organic Preparations and Procedures International

Year:

1995

Language:

english

File:

PDF, 472 KB

english, 1995

19

SYNTHESIS OF FLUORESCEIN PHOSPHATES AND SULFATES

Scheigetz, John, Gilbert, Michael, Zamboni, Robert

Journal:

Organic Preparations and Procedures International

Year:

1997

Language:

english

File:

PDF, 532 KB

english, 1997

20

Facile preparations of 4-fluororesorcinol

Bélanger, Patrice C., Lau, C. K., Williams, Haydn W. R., Dufresne, C., Scheigetz, John

Journal:

Canadian Journal of Chemistry

Year:

1988

Language:

english

File:

PDF, 286 KB

english, 1988

21

The design and synthesis of nonpeptide compounds as mimics of a conformation of methionine-enkephaline

Belanger, Patrice C., Dufresne, Claude, Scheigetz, John, Young, Robert N., Springer, James P., Dmitrienko, Gary I.

Journal:

Canadian Journal of Chemistry

Year:

1982

Language:

english

File:

PDF, 816 KB

english, 1982

22

Synthesis of Fluorescein Phosphorotriesters Using Photolabile Protecting Groups

Scheigetz, John, Roy, Bruno

Journal:

Synthetic Communications

Year:

2000

Language:

english

File:

PDF, 302 KB

english, 2000

23

Synthesis and structure-activity relationships of a novel class of 5-lipoxygenase inhibitors. 2-(Phenylmethyl)-4-hydroxy-3,5-dialkylbenzofurans: the development of L-656,224

Lau, Cheuk K., Belanger, Patrice C., Scheigetz, John, Dufresne, Claude, Williams, Haydn W. R., Maycock, Alan L., Guindon, Yvan, Bach, Thomas, Dallob, Aimee L.

Journal:

Journal of Medicinal Chemistry

Year:

1989

Language:

english

File:

PDF, 962 KB

english, 1989

24

Preparation and analgesic properties of amino acid derivatives of (-)-5,9.alpha.-diethyl-2'-hydroxybenzomorphan

Belanger, Patrice C., Scheigetz, John, Young, Robert N., Charleson, Stella E., Hudgin, Roger L., Engelhardt, Edward L.

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 456 KB

english, 1981

25

Preparation and stereochemistry of 8- and 9-hydroxy-2,5-ethano-3-benzazocines

Bélanger, Patrice C., Scheigetz, John, Young, Robert N.

Journal:

Canadian Journal of Chemistry

Year:

1983

Language:

english

File:

PDF, 351 KB

english, 1983

26

Reactions of 2-phenyl-4 H -1,3,2-benzodioxaborin, a stable ortho -quinone methide precursor

Chambers, Jeffrey D., Crawford, Jason, Williams, Haydn W. R., Dufresne, Claude, Scheigetz, John, Bernstein, Michael A., Lau, Cheuk K.

Journal:

Canadian Journal of Chemistry

Year:

1992

Language:

english

File:

PDF, 933 KB

english, 1992

27

Synthesis of 5-Methanesulfonamido-6-(2,4-Difluorophenylthio)-1-Indanone

Scheigetz, John, Zamboni, Robert, Roy, Bruno

Journal:

Synthetic Communications

Year:

1995

Language:

english

File:

PDF, 512 KB

english, 1995

28

Asymmetric Dihydroxylation of Dienes: Synthesis of Tetrols

Belley, Michel L., Hill, Bryan, Mitenko, Hugh, Scheigetz, John, Zamboni, Robert

Journal:

Year:

1996

File:

PDF, 243 KB

1996

29

Practical and Efficient Route to ( S )-γ-Fluoroleucine

Truong, Vouy Linh, Gauthier, Jacques Yves, Boyd, Michael, Roy, Bruno, Scheigetz, John

Journal:

Year:

2005

Language:

english

File:

PDF, 45 KB

english, 2005